MYP_171784
Indium In-111 Pentetreotide
Anticancer
▸
Anti-proliferative
not Standard
8 amino acids
-
contains X representing unresolved or non-standard residue
FCFWKTCX
0.00 Da
0.00
0.00
0.00
0.00
0.00
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Amino Acid Composition
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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RECORD: Rec_0009075
VERIFIED: YES
Provenance & Taxonomy
Homo sapiens [Animal]; synthetic construct [Synthetic]
Somatostatin
9606;32630
Structure & Mods
disulfide-constrained cyclic peptide [Cyclic]
mixed L/D amino-acid peptide [Mixed]
DTPA
2-aminobutane-1,3-diol
2月7日
Non-standard residues/X at 8; DTPA
Bio-Activity Profile
Diagnostic imaging
Somatostatin receptor imaging
Somatostatin receptor-positive neuroendocrine lesions
Clinical/Human: The maximum effective half-life of indium In 111 pentetreotide is 10 h.
RECORD: Rec_0405991
VERIFIED: YES
Provenance & Taxonomy
Homo sapiens [Animal]; synthetic construct [Synthetic]
Somatostatin
9606;32630
Structure & Mods
disulfide-constrained cyclic peptide [Cyclic]
mixed L/D amino-acid peptide [Mixed]
2月7日
Non-standard residues/X at 8
Bio-Activity Profile
Somatostatin receptor agonist
Antisecretory
Anti-proliferative
Human somatostatin receptors, especially SSTR2
Clinical/Human: 100 min (SC)