MYP_159311
Basic Information
D-Apidaecin-1B [1Orn,10 R], D-Api88
Anticancer
Anticancer Cytotoxic anticancer activity Cytotoxic
Antimicrobial
Antimicrobial Antibacterial
Antimicrobial Antibacterial Anti-Gram-negative
Antimicrobial Antibacterial Anti-Gram-positive
Antimicrobial Antibacterial Anti-Mycobacterium
Delivery / Targeting Barrier transport Blood-brain barrier shuttle Blood-Brain Barrier
Delivery / Targeting Drug delivery vehicle
Toxicity / Safety Blood cell toxicity Hemolysis Hemolytic
Toxicity / Safety Cytotoxicity
Toxicity / Safety Cytotoxicity Cytotoxic
Venom / Toxin General toxin Cytotoxic
Venom / Toxin General toxin Cytotoxicity
not Standard
18 amino acids
-
contains X representing unresolved or non-standard residue
Sequence
XNNRPVYIPRPRPPHPRL
Physicochemical Analysis
0.00 Da
0.00
0.00
0.00
0.00
0.00
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Residue Composition
Amino Acid Composition
Chemical Descriptors
Structural Visualization
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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Experimental Records
RECORD: Rec_0392156 VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
Synthetic designed peptide
32630
Structure & Mods
linear peptide [Linear]
noncanonical stereochemical modification [Modified]
None
Amidation
Non-standard residues/chemistry in sequence: ONNRPVYIPRPRPPHPRL
Bio-Activity Profile
Antimicrobial Antimycobacterial
Mycobacterium vaccae
MIC
RECORD: Rec_0397017 VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
synthetic linear peptide [Linear]
all-D amino-acid peptide [D]
unspecified non-canonical residue at 1
Bio-Activity Profile
Antimicrobial Antibacterial
Pseudomonas aeruginosa 61118003
1 μg/mL
MIC
RECORD: Rec_0397185 VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
synthetic linear peptide [Linear]
all-D amino-acid peptide [D]
unspecified non-canonical residue at 1
Bio-Activity Profile
Antimicrobial Antibacterial
Escherichia coli D31
64 μg/mL
MIC
RECORD: Rec_0397925 VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
synthetic linear peptide [Linear]
all-D amino-acid peptide [D]
unspecified non-canonical residue at 1
Bio-Activity Profile
Antimicrobial Antibacterial
Erwinia amylovora PMV 6076
25-50 μM
MIC
RECORD: Rec_0400536 VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
synthetic linear peptide [Linear]
all-D amino-acid peptide [D]
unspecified non-canonical residue at 1
Bio-Activity Profile
Antimicrobial Antibacterial
Escherichia coli 8474
0.5 μg/mL
MIC
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