MYP_152608
Basic Information
Dermaseptin-PP
Anticancer
Anticancer Cytotoxic anticancer activity Cytotoxic
Antimicrobial
Antimicrobial Antifungal
Toxicity / Safety Blood cell toxicity Hemolysis Hemolytic
Toxicity / Safety Cytotoxicity Cytotoxic
Venom / Toxin General toxin Cytotoxic
Wound healing/Regeneration Wound healing
Standard
26 amino acids
C123H214N32O30S
Standard
Sequence
ALWKDMLKGIGKLAGKAALGAVKTLV
Physicochemical Analysis
2653.28 Da
10.18
3.79
3.60
0.1458
0.64
0.71
0.26
-5.24
131.54
0.0385
5500.00
5500.00
The radar chart summarizes major physicochemical dimensions for quick comparison, while exact numerical values remain listed on the left.
Residue Composition
Amino Acid Composition
Chemical Descriptors
994.24
-5.29
35.0
35.0
93.0
186.0
2.0
25.0
Structural Visualization
3D PDB MODEL
Drag to rotate. Click a residue or atom to inspect it; the selected residue is highlighted in amber in the current view mode. Use the buttons to zoom.
2D CHEMICAL STRUCTURE
Drag to move
Drag to move. Use the buttons to zoom.
Experimental Records
RECORD: Rec_0186524 VERIFIED: YES
Provenance & Taxonomy
Phyllomedusa palliata [Animal]
Dermaseptin
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
APD analysis reveals that this sequence is similar (85.71%) to Dermaseptin-B3 L=A=K: 19%; G: 15%. GRAVY: 0.638; mol Wt: 2653.3; mol formula: C123H215N32O30S1; mol ex coeff: 5550. Chemical modification: Reduction of disulfide bonds and alkylation of cysteines indicate that disulfide bonds are important for peptide stability rather than activity
Bio-Activity Profile
Antimicrobial Antifungal Anticancer Wound healing
Candida albicans CYC 1467
1 μM
MIC
RECORD: Rec_0224649 VERIFIED: YES
Provenance & Taxonomy
Phyllomedusa palliata [Animal]
Dermaseptin
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
None
None
Bio-Activity Profile
Antimicrobial Anticancer Hemolytic
Horse erythrocytes: Dermaseptin-PP exhibited only a moderate hemolytic effect (<20% at 16 μM with a calculated HC50 of 38.77 μM)
RECORD: Rec_0228664 VERIFIED: YES
Provenance & Taxonomy
Phyllomedusa palliata [Animal]
Dermaseptin
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
APD analysis reveals that this sequence is similar (85.71%) to Dermaseptin-B3 L=A=K: 19%; G: 15%. GRAVY: 0.638; mol Wt: 2653.3; mol formula: C123H215N32O30S1; mol ex coeff: 5550. Chemical modification: Reduction of disulfide bonds and alkylation of cysteines indicate that disulfide bonds are important for peptide stability rather than activity
Bio-Activity Profile
Antimicrobial Antifungal Anticancer Wound healing
Pseudomonas aeruginosa ATCC 27853
2 μM
MIC
RECORD: Rec_0259843 VERIFIED: YES
Provenance & Taxonomy
Phyllomedusa palliata [Animal]
Dermaseptin
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
APD analysis reveals that this sequence is similar (85.71%) to Dermaseptin-B3 L=A=K: 19%; G: 15%. GRAVY: 0.638; mol Wt: 2653.3; mol formula: C123H215N32O30S1; mol ex coeff: 5550. Chemical modification: Reduction of disulfide bonds and alkylation of cysteines indicate that disulfide bonds are important for peptide stability rather than activity
Bio-Activity Profile
Antimicrobial Antifungal Anticancer Wound healing
Staphylococcus aureus NCTC 10788or MRSA NCTC 12493
2 μM
MIC
RECORD: Rec_0282688 VERIFIED: YES
Provenance & Taxonomy
Phyllomedusa palliata [Animal]
Dermaseptin
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
APD analysis reveals that this sequence is similar (85.71%) to Dermaseptin-B3 L=A=K: 19%; G: 15%. GRAVY: 0.638; mol Wt: 2653.3; mol formula: C123H215N32O30S1; mol ex coeff: 5550. Chemical modification: Reduction of disulfide bonds and alkylation of cysteines indicate that disulfide bonds are important for peptide stability rather than activity
Bio-Activity Profile
Antimicrobial Antifungal Anticancer Wound healing
Escherichia coli NCTC 10418
2 μM
MIC
Showing 5 records on this page · Page 2 of 4