MYP_133186
Diketopiperazine (preWH)
Anticancer
Anticancer
▸
Cytotoxic anticancer activity
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Cytotoxic
Antimicrobial
Immunology
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Immune modulation
▸
Immunomodulatory activity
Toxicity / Safety
▸
Blood cell toxicity
▸
Hemolysis
▸
Hemolytic
Toxicity / Safety
▸
Cytotoxicity
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Cytotoxic
Venom / Toxin
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General toxin
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Cytotoxic
not Standard
2 amino acids
-
contains X representing unresolved or non-standard residue
XH
0.00 Da
0.00
0.00
0.00
0.00
0.00
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Amino Acid Composition
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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RECORD: Rec_0055496
VERIFIED: YES
Provenance & Taxonomy
Synthetic construct [Synthetic]
32630
Structure & Mods
side-chain cyclized/stapled peptide [Cyclic]
canonical L-amino-acid peptide [L]
None
None
X=Prenylated-Trp
Bio-Activity Profile
Antimicrobial
Anticancer
A2780-cisR
91.7 μM
IC50
RECORD: Rec_0113741
VERIFIED: YES
Provenance & Taxonomy
Synthetic construct [Synthetic]
32630
Structure & Mods
side-chain cyclized/stapled peptide [Cyclic]
canonical L-amino-acid peptide [L]
None
None
X=Prenylated-Trp
Bio-Activity Profile
Antimicrobial
Anticancer
Cytotoxic
RECORD: Rec_0117887
VERIFIED: YES
Provenance & Taxonomy
Synthetic construct [Synthetic]
32630
Structure & Mods
side-chain cyclized/stapled peptide [Cyclic]
canonical L-amino-acid peptide [L]
None
None
X=Prenylated-Trp
Bio-Activity Profile
Antimicrobial
Anticancer
A2780
91.8 μM
IC50
RECORD: Rec_0125594
VERIFIED: NO
Provenance & Taxonomy
Bos taurus [Animal]
9913
Structure & Mods
linear peptide [Linear]
noncanonical stereochemical modification [Modified]
A1: beta-alanine
Bio-Activity Profile
Broad-spectrum activity
RECORD: Rec_0133486
VERIFIED: NO
Provenance & Taxonomy
Bos taurus [Animal]; Homo sapiens [Animal]; Ovis aries [Animal]; Equus caballus [Animal]; Rattus norvegicus [Animal]; Mus musculus [Animal]; Felis silvestris catus [Animal]; Cavia porcellus [Animal]; Balaenoptera physalus [Animal]
9913, 9606, 9940, 9796, 10116, 10090, 10141
Structure & Mods
linear peptide [Linear]
noncanonical stereochemical modification [Modified]
A1: gamma-aminobutyric acid
Bio-Activity Profile
Immunomodulatory
Showing 5 records on this page · Page 1 of 2