MYP_128984
TY027
Binding / Molecular interaction
▸
Binding activity
Neurological / Signaling
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Analgesic/opioid activity
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Analgesic
Standard
8 amino acids
C50H65N9O10S
Standard
YAGFMPLW
984.17 Da
5.52
-0.24
-0.45
-0.0301
0.76
0.20
0.65
122.88
61.25
0.3750
6990.00
6990.00
The radar chart summarizes major physicochemical dimensions for quick comparison, while exact numerical values remain listed on the left.
Amino Acid Composition
294.25
1.66
10.0
11.0
25.0
70.0
5.0
7.0
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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RECORD: Rec_0158903
VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
linear peptide [Linear]
mixed L/D amino-acid peptide [Mixed]
None
NH-[3’,5’-(CF3 )2 Bzl]
D-residue notation at positions 2; Mixed L/D stereochemistry with D-annotated positions 2
Bio-Activity Profile
Analgesic
HPLC
Rat plasma, in vitro; 17280 s
RECORD: Rec_0204851
VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
linear peptide [Linear]
mixed L/D amino-acid peptide [Mixed]
None
NH-3,5-Bzl(CF3)2
D-residue notation at positions 2; Mixed L/D stereochemistry with D-annotated positions 2
Bio-Activity Profile
Receptor-binding
MVD
0.015±0.002 μM
IC50
Rat plasma, in vitro; 17280 s
RECORD: Rec_0301430
VERIFIED: YES
Provenance & Taxonomy
synthetic construct [Synthetic]
32630
Structure & Mods
linear peptide [Linear]
mixed L/D amino-acid peptide [Mixed]
None
O-[3’,5’-(CF3 )2 Bzl]
D-residue notation at positions 2; Mixed L/D stereochemistry with D-annotated positions 2
Bio-Activity Profile
Analgesic
HPLC
Rat plasma, in vitro; 86400 s