MYP_089459
Diketopiperazine LR [R2 modified]
Anticancer
Anticancer
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Cytotoxic anticancer activity
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Cytotoxic
Antimicrobial
Antimicrobial
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Antifungal
Antiparasitic
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Antiprotozoal
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Antimalarial
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Anti-Plasmodium
Antiparasitic
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General antiparasitic
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Antiparasitic
Enzyme modulation
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Enzyme inhibition
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ACE inhibition
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ACE inhibitory
Enzyme modulation
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Enzyme inhibition
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Protease inhibition
Other / Curated residual function label
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Generic enzyme inhibition annotation
Toxicity / Safety
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Blood cell toxicity
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Hemolysis
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Hemolytic
Toxicity / Safety
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Cytotoxicity
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Cytotoxic
Venom / Toxin
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General toxin
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Cytotoxic
not Standard
2 amino acids
-
contains X representing unresolved or non-standard residue
LX
0.00 Da
0.00
0.00
0.00
0.00
0.00
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Amino Acid Composition
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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RECORD: Rec_0000685
VERIFIED: YES
Provenance & Taxonomy
Bacillus cereus [Bacterium]
Structure & Mods
head-to-tail cyclic peptide [Cyclic]
mixed L/D amino-acid peptide [Mixed]
R2: D-arg
Bio-Activity Profile
Antimicrobial
Antifungal
Candida albicans
8 μg/mL
MIC
RECORD: Rec_0101531
VERIFIED: YES
Provenance & Taxonomy
Homo sapiens [Animal]
9606
Structure & Mods
linear peptide [Linear]
noncanonical stereochemical modification [Modified]
P2: hydroxyproline
Bio-Activity Profile
Enzyme inhibitory
ACE inhibitory
Angiotensin-converting enzyme
3462.1 ± 1012.2 μM
IC50
RECORD: Rec_0147475
VERIFIED: YES
Provenance & Taxonomy
not reported [other]
Structure & Mods
linear peptide [Linear]
mixed L/D amino-acid peptide [Mixed]
Z=benzyloxycarbonyl
Al=aldehyde
HPhe=homophenylalanine
Bio-Activity Profile
Antiparasitic
Antimicrobial
Antiplasmodial
Cysteine protease inhibitor
RECORD: Rec_0150480
VERIFIED: YES
Provenance & Taxonomy
not reported [other]
Structure & Mods
linear peptide [Linear]
mixed L/D amino-acid peptide [Mixed]
Mu=Morpholine urea
CH2F
HPhe=Homophenylalanine
Bio-Activity Profile
Antiparasitic
Antimicrobial
Antiplasmodial
Cysteine protease inhibitor
RECORD: Rec_0203255
VERIFIED: YES
Provenance & Taxonomy
Fungi [Fungus]
Structure & Mods
linear peptide [Linear]
canonical L-amino-acid peptide [L]
None
None
Bio-Activity Profile
Antimicrobial
Anticancer
Not available
Showing 5 records on this page · Page 1 of 3