MYP_030015
Basic Information
Endothelin-1
Cardiovascular
Cardiovascular Vascular tone modulation Vasoactive peptide
Cardiovascular Vascular tone modulation Vasoconstrictor activity
Enzyme modulation Enzyme inhibition ACE inhibition ACE inhibitory
Hormonal / Endocrine Hormone peptide
Neurological / Signaling Neuromuscular and muscle activity Myotropic activity
Regulatory peptide Biological modulation
Standard
21 amino acids
C110H165N25O32S4
Standard
Sequence
CSCSSLLDKECVYFCHLDIIW
Physicochemical Analysis
2477.90 Da
4.54
-2.19
-2.51
-0.1043
0.72
0.30
0.26
59.44
106.67
0.1429
6990.00
7240.00
The radar chart summarizes major physicochemical dimensions for quick comparison, while exact numerical values remain listed on the left.
Residue Composition
Amino Acid Composition
Chemical Descriptors
908.63
-5.50
36.0
35.0
78.0
171.0
5.0
20.0
Structural Visualization
3D PDB MODEL
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2D CHEMICAL STRUCTURE
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Experimental Records
RECORD: Rec_0108691 VERIFIED: NO
Provenance & Taxonomy
Felis catus [Animal]
Endothelin/sarafotoxin
9685
Structure & Mods
disulfide-constrained cyclic peptide [Cyclic]
canonical L-amino-acid peptide [L]
1-15; 3-11
Bio-Activity Profile
Vasoactive Hormone
RECORD: Rec_0250878 VERIFIED: NO
Provenance & Taxonomy
Felis catus [Animal]
Endothelin
9685
Structure & Mods
disulfide-constrained peptide [Cyclic]
canonical L-amino-acid peptide [L]
1-15; 3-11
Bio-Activity Profile
Hormone Endocrine Vasoactive Vasoconstrictor Cardiovascular Myotropic Receptor modulation ACE inhibitory
Mammalian: 1.2 hour; Yeast: >20 hour; E. coli: >10 hour
RECORD: Rec_0284408 VERIFIED: NO
Provenance & Taxonomy
Felis catus [Animal]
Endothelin
9685
Structure & Mods
disulfide-constrained peptide [Cyclic]
canonical L-amino-acid peptide [L]
1-15; 3-11
Bio-Activity Profile
Hormone Endocrine Vasoactive Vasoconstrictor Cardiovascular Myotropic Receptor modulation ACE inhibitory
glomerular mesangial cells
Mammalian: 1.2 hour; Yeast: >20 hour; E. coli: >10 hour