ASSAY RECORD
Results
Showing up to 20 records.
| NO. | RECORD ID | NAME | SEQUENCE | SOURCE ORGANISM | FUNCTION CATEGORY | TARGET ORGANISM | ACTIVITY | ASSAY METHOD | PMID | PATENT NO | VERIFICATION STATUS |
|---|---|---|---|---|---|---|---|---|---|---|---|
| 428081 | Rec_0431337 | Extended structure of citidine deaminase domain of APOBEC3G |
GPLGSPGFEILRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
19389408 | - |
YES |
| 428082 | Rec_0431338 | The Crystal Structure of the Anti-Viral APOBEC3G Catalytic Domain |
GPLGSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVLLNQRRGFLCNQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIFTARIYDDQGRCQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGCPFQPWDGLDEHSQDLSGRLRAILQ |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
18849968 | - |
YES |
| 428083 | Rec_0431339 | Solution structure of peptide H30 by Nuclear Magnetic Resonance Spectroscopy |
GAICHPVFCPRRYKQIGTCGLPGTKCCKKP |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
- | - |
YES |
| 428084 | Rec_0431340 | Structure based design of RIP1 kinase inhibitors |
GGSGQPDMSLNVIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELREVDGTAKKNGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE |
Homo sapiens [other] |
Cell-penetrating |
- |
- | X-ray |
29485864 | - |
YES |
| 428085 | Rec_0431341 | 1.20 A resolution structure of Norovirus 3CL protease in complex with a triazole-based macrocyclic (17-mer) inhibitor |
MHHHHHHAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQAGEGETALE |
Norwalk virus [other] |
Antiviral |
- |
- | X-ray |
27235842 | - |
YES |
| 428086 | Rec_0431342 | Solution structure of chicken Engrailed 2 homeodomain |
GPMASDKRPRTAFTAEQLQRLKAEFQTNRYLTEQRRQSLAQELGLNESQIKIWFQNKRAKIKKATQA |
GALLUS GALLUS [other] |
Cell-penetrating |
- |
- | NMR |
23931315 | - |
YES |
| 428087 | Rec_0431343 | Crystal structure of antibody scFv against M2e Influenza peptide |
MAEVQLLESGGGLVQPGGSLRLSCAASGFTFSSYAMSWVRQAPGKGLEWVSTILQHGQRTLYADSVKGRFTISRDNSKNTLYLQMNSLRAEDTAVYYCAKNRAVFDYWGQGTLVTVSSGGGGSGGGGSGGGGSTDIQMTQSPSSLSASVGDRVTITCRASQSISSYLNWYQQKPGKAPKLLIYTASTLQSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQYRQRPPTFGQGTKVEIKRAAALEHHHHHH |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
37491224 | - |
YES |
| 428088 | Rec_0431344 | Crystal Structure of N-terminal Human IFIT1 |
DHQVKDSLEQLRCHFTWELSIDDDEMPDLENRVLDQIEFLDTKYSVGIHNLLAYVKHLKGQNEEALKSLKEAENLMQEEHDNQANVRSLVTWGNFAWMYYHMGRLAEAQTYLDKVENICKKLSNPFRYRMECPEIDCEEGWALLKCGGKNYERAKACFEKVLEVDPENPESSAGYAISAYRLDGFKLATKNHKPFSLLPLRQAVRLNPDNGYIKVLLALKLQDEGQEAEGEKYIEEALANMSSQTYVFRYAAKFYRRKGSVDKALELLKKALQ |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
23334420 | - |
YES |
| 428089 | Rec_0431345 | HIV-1 protease triple mutants V32I, I47V, V82I with GRL-011-11A (a methylamine bis-Tetrahydrofuran P2-Ligand, sulfonamide isostere derivate) |
PQITLWKRPLVTIKIGGQLKEALLDTGADDTIIEEMSLPGRWKPKMVGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPINIIGRNLLTQIGATLNF |
Human immunodeficiency virus 1 [other] |
Antiviral |
- |
- | X-ray |
31092330 | - |
YES |
| 428090 | Rec_0431346 | Structure of Enterovirus A71 3C protease |
MGPSLDFALSLLRRNIRQVQTDQGHFTMLGVRDRLAVLPRHSQPGKTIWVEHKLINILDAVELVDEQGVNLELTLVTLDTNEKFRDITKFIPENISAASDATLVINTEHMPSMFVPVGDVVQYGFLNLSGKPTHRTMMYNFPTKAGQCGGVVTSVGKVIGIHIGGNGRQGFCAGLKRSYFASEQLEHHHHHH |
Enterovirus [other] |
Antiviral |
- |
- | X-ray |
- | - |
YES |
| 428091 | Rec_0431347 | Crystal structure of APOBEC3F-CD1 |
GPGGSGGMKPHFRNTVERMDRDTFSYNFYNEPILARRNTVWLCYEVKTKGPSRPRLDAKIFRGQVYSQPEHHAEMCFLSWFCGNQLPADKCFQITWFVSWTPCPDCVAKLAEFLAEHPNVTLTISAARLYYYSERDYRRALCRLSQAGARVKIMDDEEFAYCWENFVDSEGQPFMPWYKFDDNYAFLHRTLKEILRN |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
41207371 | - |
YES |
| 428092 | Rec_0431348 | Structural basis of oligomerisation in the MxA stalk |
EDENEKMFFLIDKVNAFNQDITALMQGEETVGEEDIRLFTRLRHEFHKWSTIIENNFQEGHKILSRKIQKFENQYRGRELPGFVNYRTFETIVKQQIKALEEPAVDMLHTVTDMVRLAFTDVSIKNFEEFFNLHRTAKSKIEDIRAEQEREGEKLIRLHFQMEQIVYCQDQVYRGALQKVREKELEEEKKKKSWDFGAFQSSSATDSSMEEIFQHLMAYHQEASKRISSHIPLIIQFFMLQTYGQQLQKAMLQLLQDKDTYSWLLKERSDT |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
20428112 | - |
YES |
| 428093 | Rec_0431349 | First-In-Class Small Molecule Inhibitors of the Single-strand DNA Cytosine Deaminase APOBEC3G |
GPLGSPEFELGTTEILRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
22181350 | - |
YES |
| 428094 | Rec_0431350 | First-In-Class Small Molecule Inhibitors of the Single-strand DNA Cytosine Deaminase APOBEC3G |
GPLGSPEFELGTTEILRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRCQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQ |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
22181350 | - |
YES |
| 428095 | Rec_0431351 | C-TERMINAL DOMAIN OF INFLUENZA POLYMERASE PA SUBUNIT AND OPTIMIZED SMALL PEPTIDE INHIBITOR |
DYNPYLLFLK |
synthetic construct [other] |
Antiviral |
- |
- | X-ray |
33166574 | - |
YES |
| 428096 | Rec_0431352 | CRYSTAL STRUCTURE OF APOBEC3G CATALYTIC DOMAIN COMPLEX WITH SUBSTRATE SSDNA |
AATCCCAAA |
synthetic construct [other] |
Antiviral |
- |
- | X-ray |
29941968 | - |
YES |
| 428097 | Rec_0431353 | CRYSTAL STRUCTURE OF APOBEC3G CATALYTIC DOMAIN COMPLEX WITH SUBSTRATE SSDNA |
GPLGSEILRHSMDPATFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLAQRRGFLANQAKHKHGFLEGRHAALCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDKGRAAEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
29941968 | - |
YES |
| 428098 | Rec_0431354 | Three-Dimensional Structures of Cm-p1 |
SRSELIVHQRX |
Cenchritis muricatus [other] |
Antifungal |
- |
- | NMR |
- | - |
YES |
| 428099 | Rec_0431355 | Vaccatide: Antifungal Glutamine-rich 8C-Hevein-like Peptide, vH1 |
FQCGRQAGGARCSNGLCCSQFGYCGSTPPYCGAGQCQSQC |
Vaccaria hispanica [other] |
Antifungal |
- |
- | NMR |
28680440 | - |
YES |
| 428100 | Rec_0431356 | Chickpea (Cicer arientinum) nodule-specific cysteine-rich peptide NCR13: Solution NMR structure of the isomer with C4:C10, C15:C30, and C23:C28 disulfide bonds |
ATKPCQSDKDCKKFACRKPKVPKCINGFCKCVR |
Cicer arientinum [other] |
Antifungal |
- |
- | NMR |
39621770 | - |
YES |