ASSAY RECORD
Results
Showing up to 20 records.
| NO. | RECORD ID | NAME | SEQUENCE | SOURCE ORGANISM | FUNCTION CATEGORY | TARGET ORGANISM | ACTIVITY | ASSAY METHOD | PMID | PATENT NO | VERIFICATION STATUS |
|---|---|---|---|---|---|---|---|---|---|---|---|
| 424401 | Rec_0431322 | NMR structure analysis of the Penetratin conjugated Gas (374-394) peptide |
RQIKIWFQNRRMKWKKRVFNDARDIIQRMHLRQYELL |
- |
Cell-penetrating |
- |
- | NMR |
17348636 | - |
YES |
| 424402 | Rec_0431323 | Structure of DK17 in POPC:POPG:Cholesterol:GM1 LUVS |
DRQIKIWFQNRRMKWKK |
Drosophila melanogaster [other] |
Cell-penetrating |
- |
- | NMR |
27532224 | - |
YES |
| 424403 | Rec_0431324 | Crystal structure of MCL-1 in complex with a neutralizing Alphabody CMPX-383B |
GSHMGSDELYRQSLEIISRYLREQATGAKDTKPMGRSGATSRKALETLRRVGDGVQRNHETAFQGMLRKLDIKNEDDVKSLSRVMIHVFSDGVTNWGRIVTLISFGAFVAKHLKTINQESCIEPLAESITDVLVRTKRDWLVKQRGWDGFVEFFHVEDLEGG |
Homo sapiens [other] |
Cell-penetrating |
- |
- | X-ray |
33771865 | - |
YES |
| 424404 | Rec_0431325 | Crystal structure of MCL-1 in complex with a neutralizing Alphabody CMPX-383B |
GSHMSTEQIQKRTAAIQKRIAAIQKRIYAMTASGGAGAAGAGAGMSIEEITKQIAAIQLRIVGDQVQIAYQTASGAGAGAGGMSTEEIQKQIAAIETQICKIEAAIELKEAGITSDFYFELINKAKTCEGVEALKEHILAAHT |
synthetic construct [other] |
Cell-penetrating |
- |
- | X-ray |
33771865 | - |
YES |
| 424405 | Rec_0431326 | Crystal structure of SARS-CoV-2 main protease in complex with Mp-4L2 |
YNLFQRTDWTTQYXGX |
synthetic construct [other] |
Cell-penetrating |
- |
- | X-ray |
- | - |
YES |
| 424406 | Rec_0431327 | Crystal structure of SARS-CoV-2 main protease in complex with Mp-4D7 |
YVTFHTTTPFLPPXGX |
synthetic construct [other] |
Cell-penetrating |
- |
- | X-ray |
- | - |
YES |
| 424407 | Rec_0431328 | CRYSTAL STRUCTURE OF RIP1 KINASE BOUND TO INHIBITOR |
GGSGQPDMSLNVIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELREVDGTAKKNGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDLTEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE |
Homo sapiens [other] |
Cell-penetrating |
- |
- | X-ray |
29485864 | - |
YES |
| 424408 | Rec_0431329 | I5R8 Mastoparano is a peptide synthetic, modified of Mastoparano (extracted from wasp venom) |
INLKILARLAKKILX |
Vespula lewisii [other] |
Antiviral |
- |
- | NMR |
- | - |
YES |
| 424409 | Rec_0431330 | Crystal structure of human Shiftless (SFL) containing phosphorylation sites Ser249, Thr250, Thr253 and Ser256 |
GSQEGVELEKSVRRLREKFHGKVSSKKAGALMRKFGSDHTGVGRSIVYGVKQKDGQELSNDLDAQDPPEDMKQDRDIQAVATSLLPLTEANLRMFQRAQDDLIPAVDRQFACSSCDHVWWRRVPQRKEVSRCRKCRKRYEPVPADKMWGLAEFHCPKCRHNFRGWAQMGSPSPCYGCGFPVYPTRILPPRWDRDPDRRSTHTHSCSAADCYNRREPHVPGTSCAHPKSRKQNHLPKVLHPSNPHISSGSTVATCLSQGGLLEDLDNLILEDLKEEEEEEEEVEDEEGGPRE |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
41417896 | - |
YES |
| 424410 | Rec_0431331 | Influenza polymerase A C-terminal domain of PA subunit with optimized small peptide inhibitor |
DYNPYLLYLK |
synthetic construct [other] |
Antiviral |
- |
- | X-ray |
36265804 | - |
YES |
| 424411 | Rec_0431332 | Crystal structure of beta-2 microglobulin (beta2m) of Bat (Pteropus Alecto) |
EPRTPKIQVYSRHPAENGKPNYLNCYVYGFHPPQIEIDLLKNGQKMKTEQSDLSFSKDWSFYLLVHTDFTPSTVDEYSCRVNHSSLAAPHMVKWDRNNT |
Pteropus alecto [other] |
Antiviral |
- |
- | X-ray |
31498797 | - |
YES |
| 424412 | Rec_0431333 | Crystal structure of antibody scFv against M2e Influenza peptide |
MAEVQLLESGGGLVQPGGSLRLSCAASGFTFSSYAMSWVRQAPGKGLEWVSGISQLGGYTGYAGSVKGRFTISRDNSKNTLYLQMNSLRAEDTAVYYCAKNRATFDYWGQGTLVTVSSGGGGSGGGGSGGGGSTDIQMTQSPSSLSASVGDRVTITCRASQSISSYLNWYQQKPGKAPKLLIYAASHLQSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQSQHKPLTFGQGTKVEIKRAAALEHHHHHH |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
37491224 | - |
YES |
| 424413 | Rec_0431334 | Crystal structure of CTSB in complex with K777 |
KLPASFDAREQWPQCPTIKEIRDQGSCGSCWAFGAVEAISDRICIHTNAHVSVEVSAEDLLTCCGSMCGDGCNGGYPAEAWNFWTRKGLVSGGLYESHVGCRPYSIPPCEHHVNGSRPPCTGEGDTPKCSKICEPGYSPTYKQDKHYGYNSYSVSNSEKDIMAEIYKNGPVEGAFSVYSDFLLYKSGVYQHVTGEMMGGHAIRILGWGVENGTPYWLVANSWNTDWGDNGFFKILRGQDHCGIESEVVAGIPRTD |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
37990007 | - |
YES |
| 424414 | Rec_0431335 | Solution structure of C-terminal domain of APOBEC3G |
GPLGSPEFDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
18288108 | - |
YES |
| 424415 | Rec_0431336 | Structure, interaction, and real-time monitoring of the enzymatic reaction of wild type APOBEC3G |
HMLRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVLLNQRRGFLCNQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIFTARIYDDQGRCQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGCPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
19153609 | - |
YES |
| 424416 | Rec_0431337 | Extended structure of citidine deaminase domain of APOBEC3G |
GPLGSPGFEILRHSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVKLNQRRGFLANQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIKTARIYDDQGRAQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGAPFQPWDGLDEHSQDLSGRLRAILQNQEN |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
19389408 | - |
YES |
| 424417 | Rec_0431338 | The Crystal Structure of the Anti-Viral APOBEC3G Catalytic Domain |
GPLGSMDPPTFTFNFNNEPWVRGRHETYLCYEVERMHNDTWVLLNQRRGFLCNQAPHKHGFLEGRHAELCFLDVIPFWKLDLDQDYRVTCFTSWSPCFSCAQEMAKFISKNKHVSLCIFTARIYDDQGRCQEGLRTLAEAGAKISIMTYSEFKHCWDTFVDHQGCPFQPWDGLDEHSQDLSGRLRAILQ |
Homo sapiens [other] |
Antiviral |
- |
- | X-ray |
18849968 | - |
YES |
| 424418 | Rec_0431339 | Solution structure of peptide H30 by Nuclear Magnetic Resonance Spectroscopy |
GAICHPVFCPRRYKQIGTCGLPGTKCCKKP |
Homo sapiens [other] |
Antiviral |
- |
- | NMR |
- | - |
YES |
| 424419 | Rec_0431340 | Structure based design of RIP1 kinase inhibitors |
GGSGQPDMSLNVIKMKSSDFLESAELDSGGFGKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELREVDGTAKKNGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE |
Homo sapiens [other] |
Cell-penetrating |
- |
- | X-ray |
29485864 | - |
YES |
| 424420 | Rec_0431341 | 1.20 A resolution structure of Norovirus 3CL protease in complex with a triazole-based macrocyclic (17-mer) inhibitor |
MHHHHHHAPPTLWSRVTKFGSGWGFWVSPTVFITTTHVVPTGVKEFFGEPLSSIAIHQAGEFTQFRFSKKMRPDLTGMVLEEGCPEGTVCSVLIKRDSGELLPLAVRMGAIASMRIQGRLVHGQSGMLLTGANAKGMDLGTIPGDCGAPYVHKRGNDWVVCGVHAAATKSGNTVVCAVQAGEGETALE |
Norwalk virus [Virus] |
Antiviral |
- |
- | X-ray |
27235842 | - |
YES |