ASSAY RECORD
Results
Showing up to 20 records.
| NO. | RECORD ID | NAME | SEQUENCE | SOURCE ORGANISM | FUNCTION CATEGORY | TARGET ORGANISM | ACTIVITY | ASSAY METHOD | PMID | PATENT NO | VERIFICATION STATUS |
|---|---|---|---|---|---|---|---|---|---|---|---|
| 420381 | Rec_0433039 | S25 |
KKAAASAAAAASAAWAASAAAKKKK |
synthetic construct [Synthetic] |
Antimicrobial, Antibacterial |
Staphylococcus epidermidis C621 |
>64 μM | MIC |
- | US 2004/0235745 A1 |
YES |
| 420382 | Rec_0433040 | PF-525 |
KFSDQIDKGQDALKDKLGDL |
synthetic construct [Synthetic] |
Antimicrobial, Antibacterial |
Streptococcus pneumoniae |
50 μM | MIC |
- | US 2010/0184681 A1 |
YES |
| 420383 | Rec_0433041 | Bacteriocin Enterocin 1071 subunit beta [K4G] |
GPGGWLPWLQPAYDFVTGLAKGIGKEGNKNKWKNV |
synthetic construct [Synthetic] |
Antimicrobial, Antibacterial |
Enterococcus faecalis NCDO 581 |
1.0±0.3 nM | MIC (with Ent-α, 1:1 complementary peptide mixture) |
17337546 | - |
YES |
| 420384 | Rec_0433042 | Bacteriocin Enterocin 1071 subunit beta [K4G] |
GPGGWLPWLQPAYDFVTGLAKGIGKEGNKNKWKNV |
synthetic construct [Synthetic] |
Antimicrobial, Antibacterial |
Enterococcus faecalis LMGT-2333 |
1.0±0.3 nM | MIC (with Ent-α, 1:1 complementary peptide mixture) |
17337546 | - |
YES |
| 420385 | Rec_0433043 | YSA (EphA2-targeting peptide) |
YSAYPDSVPMMSK |
synthetic construct [Synthetic] |
Targeting, Drug delivery, Anticancer |
EphA2 receptor; MDA-MB-231 cells; HUVEC |
- | EphA2-targeted cellular uptake/binding assay; in vivo tumor-targeting study |
26004003 | - |
YES |
| 420386 | Rec_0433044 | thionin Osthi1 |
KSCCPSTTARNVYNSCRFAGGSRDTCAKLSGCKIVDGNCKPPYVH |
Oryza sativa subsp. japonica [Plant] |
Antimicrobial |
- |
- | Qualitative antimicrobial activity assay |
- | - |
YES |
| 420387 | Rec_0433045 | S. caprae AIP+1 |
GYSTCSYYF |
synthetic construct [Synthetic] |
Quorum Sensing Inhibition, Cell-Cell Communication |
Staphylococcus aureus agr type I reporter |
0.83 nM | agr P3-YFP reporter assay (IC50) |
29199097 | - |
YES |
| 420388 | Rec_0433046 | Allatostatin C (ScypaAST-C) |
QIRYHQCYFNPISCF |
Scylla paramamosain [Animal] |
Neuropeptide, Receptor agonist, Ecdysone biosynthesis inhibitor |
Scylla paramamosain C-type allatostatin receptor (ScypaAST-CR); HEK293T cells |
1 μM | cAMP luciferase receptor activation assay |
- | - |
YES |
| 420389 | Rec_0433047 | M-poneritoxin-Nc2a (M-PONTX-Nc2a) (Poneratoxin) (Ponericin Nc2a) |
FVKELWDKVKKMGSAAWSAAKGAFA |
Neoponera commutata [Animal] |
Insecticidal, Toxin |
Lucilia cuprina |
>100 nmol/g | LD50 (24 h lethality) |
34302796 | - |
YES |
| 420390 | Rec_0433048 | M-poneritoxin-Nc2a (M-PONTX-Nc2a) (Poneratoxin) (Ponericin Nc2a) |
FVKELWDKVKKMGSAAWSAAKGAFA |
Neoponera commutata [Animal] |
Hemolytic, Cytotoxic |
human red blood cells |
>250 μM | HC50 / Hemolysis |
34302796 | - |
YES |
| 420391 | Rec_0433049 | M-poneritoxin-Nc2a (M-PONTX-Nc2a) (Poneratoxin) (Ponericin Nc2a) |
FVKELWDKVKKMGSAAWSAAKGAFA |
Neoponera commutata [Animal] |
Cytotoxic |
HEK293 cells |
48.2-56.9 μM | CC50 |
34302796 | - |
YES |
| 420392 | Rec_0433050 | Kentsin |
TPRK |
Mesocricetus auratus [Animal] |
Gastrointestinal motility regulator, Opioid-like activity |
fasted dog antral motility |
51.2 % | Antral motility index inhibition |
4043221 | - |
YES |
| 420393 | Rec_0433051 | Kentsin |
TPRK |
Mesocricetus auratus [Animal] |
Gastrointestinal motility regulator, Opioid-like activity |
fasted dog antral motility |
76.1 % | Antral motility index inhibition |
4043221 | - |
YES |
| 420394 | Rec_0433052 | Ω17 |
RKKAIKLVKKLVKKLKKALK |
synthetic construct [Synthetic] |
Antimicrobial, Antibacterial, Anti-Gram-negative |
Escherichia coli |
2 mg/L | MBC50 |
31355341 | - |
YES |
| 420395 | Rec_0433053 | Alpha-mammal toxin Ts2 (P-Mice-beta* NaTx5.1), (Tityustoxin II), (Toxin II), (TsTX-II), (Tst2), (Toxin T1-IV), (TsTX III-8), (TsTX-III) |
KEGYAMDHEGCKFSCFIRPAGFCDGYCKTHLKASSGYCAWPACYCYGVPDHIKVWDYATNKC |
Tityus serrulatus [Animal] |
Neurotoxin, Sodium-channel modulator |
voltage-gated sodium channel NaV1.6 |
35±6 % | Electrophysiology: non-inactivating current at 1 μM Ts2 |
- | - |
YES |
| 420396 | Rec_0433054 | Alpha-mammal toxin Ts2 (P-Mice-beta* NaTx5.1), (Tityustoxin II), (Toxin II), (TsTX-II), (Tst2), (Toxin T1-IV), (TsTX III-8), (TsTX-III) |
KEGYAMDHEGCKFSCFIRPAGFCDGYCKTHLKASSGYCAWPACYCYGVPDHIKVWDYATNKC |
Tityus serrulatus [Animal] |
Neurotoxin, Sodium-channel modulator |
voltage-gated sodium channel NaV1.7 |
33±4 % | Electrophysiology: non-inactivating current at 1 μM Ts2 |
- | - |
YES |
| 420397 | Rec_0433055 | MFLG |
MFLG |
synthetic construct [Synthetic] |
Antioxidant |
- |
- | ORAC antioxidant assay |
33336193 | - |
YES |
| 420398 | Rec_0433056 | MFLG |
MFLG |
synthetic construct [Synthetic] |
ACE inhibitory, Antihypertensive |
angiotensin-converting enzyme (ACE) |
70 μM | IC50 (ACE inhibition assay) |
39942857 | - |
YES |
| 420399 | Rec_0433057 | HH969 (SEQ ID NO:969) |
IFKWFYRRK |
synthetic construct [Synthetic] |
- |
Pseudomonas aeruginosa H1001 |
- | Luminescence-based antimicrobial screening of cellulose-bound peptides |
- | US 9017656 B2 |
YES |
| 420400 | Rec_0433058 | RKSSK (IL-1Ra N-terminal peptide) |
RKSSK |
synthetic construct [Synthetic] |
Immunomodulatory, Immunosuppressive |
BALB/c mouse humoral and cellular immune response |
- | Delayed-type hypersensitivity (DTH) and plaque-forming cell (PFC) assays in vivo |
9437498 | - |
YES |